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抑制剂激活剂等> 蛋白翻译、折叠和降解> Ubiquitin/Proteasome
MG-132 (Proteasome抑制剂)
产品编号: S1748-5mg
产品包装:5mg
选择包装
价格: ¥ 415.00
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产品编号 产品名称 产品包装 产品价格
S1748-1mg MG-132 (Proteasome抑制剂) 20mg/ml×0.05ml 325.00元
S1748-5mg MG-132 (Proteasome抑制剂) 5mg 415.00元
S1748-25mg MG-132 (Proteasome抑制剂) 25mg 1461.00元

MG-132也写作MG132,也称Z-LLL-CHO,Z-Leu-Leu-Leu-CHO,Z-Leu-Leu-Leu-al或Carbobenzoxy-L-leucyl-L-leucyl-L-leucinal,是一种常用的Proteasome抑制剂,即蛋白酶体抑制剂。MG-132可以通透细胞,选择性抑制Proteasome,Ki=4nM。可以激活JNK1并抑制NF-κB的激活(IC50=3μM)。在10μM时可以诱导PC12细胞产生neurite outgrowth。
MG-132分子量为475.62,分子式为C26H41N3O5,CAS Number:133407-82-6。本产品纯度大于99%。
本MG-132为进口分装,其中20mg/ml包装产品用DMSO配制,共0.05ml。5mg和25mg包装为粉末装。
包装清单:

产品编号 产品名称 包装
S1748-1mg MG-132 (Proteasome抑制剂) 20mg/ml×0.05ml
S1748-5mg MG-132 (Proteasome抑制剂) 5mg
S1748-25mg MG-132 (Proteasome抑制剂) 25mg
说明书 1份

保存条件:
-20℃避光保存,半年有效。
注意事项:
本MG-132在4℃、冰浴等较低温度情况下会凝固而粘在离心管管底、管壁或管盖内,可以20-25℃水浴温育片刻至全部融解后使用。
本产品仅限于专业人员的科学研究用,不得用于临床诊断或治疗,不得用于食品或药品,不得存放于普通住宅内。
为了您的安全和健康,请穿实验服并戴一次性手套操作。

使用说明:

1. MG-132常见使用浓度范围为1-50μM。具体的最佳工作浓度请参考相关文献,或根据实验目的,以及所培养的特定细胞和组织,通过实验进行摸索和优化。

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